発表論文(2001年以前)及び総説・単行書・教科書

 

2001

 

1.        Songkram, C.; Takaishi, K.; Yamaguchi, K.; Kagechika, H.; Endo, Y.*

Structures of Bis- and Tris(2-phenyl-o-carboran-1-yl)benzenes. Construction of Three-dimensional Structures Converted from Planar Arylacetylenic Arrays

         Tetrahedron Lett., 2001, 42, 6365-6368.

 

2.        Endo, Y.*; Taoda, Y.,

Electronic Effects of Icosahedral Carboranes: Kinetic Evidence for Interaction between Boron Atom and Nucleophile on the Solvolysis of (o-Carboranyl)benzyl Tosylates.

Tetrahedron Lett., 2001, 42, 6327-6331.

 

3.        Yamamoto, K.; Endo, Y.*

Utility of Boron Clusters for Drug Design. Hansch-Fujita Hydrophobic Parameters p of Dicarba-closo-dodecaboranyl Groups.

BioMed. Chem. Lett., 2001, 11, 2389-2392.

 

4.        Songkram, C.; Yamasaki, R.; Takaishi, K.; Yamaguchi, K.; Kagechika, H.; Endo, Y.*

Molecular Construction Based on Icosahedral Carboranes and Aromatic Urea Groups. A New Type of Carboracycles.

Tetrahedron Lett., 2001, 42, 5913-5916.

 

5.        Sou, S.; Takahashi, H.; Yamasaki, R.; Kagechika, H.; Endo, Y.; Hashimoto, Y.,

a-Glucosidase Inhibitors with 4,5,6,7-Tetrachlorophtalimide Skeleton with a Cycloalkyl or Dicarba-closo-dodecaborane.

Chem. Pharm. Bull., 2001, 49, 791-793.

 

6.        Endo, Y.*; Iijima, T.; Yamakoshi, Y., Fukasawa, H.; Miyaura, C.; Inada, M.; Kubo, A.; Itai, A.

Potent Estrogen Agonists Based on Carborane as a Hydrophobic Skeletal Structure. A New Medicinal Application of Boron Clusters.

Chemistry and Biology, 2001, 8, 341-355.

 

7.        Endo, Y.*; Iijima, T.; Yaguchi, K.; Kawachi, E.; Kagechika, H.,

Medicinal Application of Dicarba-closo-dodecaboranes. Relation between Retinoidal Activity and Conformation of Two Aromatic Nuclei.

BioMed. Chem. Lett., 2001, 11, 1307-1311.

 

2000

 

8.        Fukasawa, H.; Yamaguchi, M.; Hashimoto, Y.; Endo, Y.; Shudo, K.

Enhancing Effect of Tumor Promoters, Phorbol Esters and Teleocidins, on Nuclear Receptor-mediated Transcription.

Biol. Pharm. Bull., 2000, 23, 1414-1417.

 

9.        Songkram, C.; Tanatani, A.; Yamasaki, R.; Yamaguchi, K.; Kagechika, H.; Endo, Y*.,

Structures of N, N’-Bis(1,2-dicarba-closo-dodecaboran-1-yl)phenylureas. Building Blocks for Carborane Containing Macromolecules.

Tetrahedron Lett., 2000, 41, 7065-7070.

 

10.    Mayumi, S.; Azuma, A.; Kobayashi, H.; Sodeoka, M.; Yano, K.; Sugimoto, S.; Endo, Y.; Hashimoto, Y.

Identification of Protein Disulfide Isomerase as a Phorbol ester-binding Protein.

Biol. Pharm.Bull., 2000, 23, 1111-1113.

 

11.    Endo, Y.*; Yaguchi, K.; Kawachi, E.; Kagechika, H.,

Polymethylcarborane as a Novel Bioactive Moiety: derivatives with Potent Retinoid Antagonistic Activity.

BioMed. Chem. Lett., 2000, 10, 1733-1736.

 

12.    Tsuji, M.; Koiso, Y.; Takahashi, H; Hashimoto, Y.; Endo, Y.

Modulators of Tumor Necrosis Factor a Production Bearing Dicarba-closo-dodecaborane as a Hydrophobic Pharmacophore.

Biol. Pharm. Bull., 2000, 23, 513-516.

 

13.    Endo, Y.*; Sawabe, T., Taoda, Y.

Electronic Effects of Dicarba-closo-dodecaboranes. Retentive Solvolysis of (1,2-Dicarba-closo-dodeca-boran-1yl)benzyl p-Toluenesulfonates.

J. Am. Chem. Soc., 2000, 122, 180-181.

 

14.    Endo, Y.*; Yoshimi, T.; Yamakoshi, Y.

New Estrogen Antagonists Bearing Dicarba-closo-dodecaborane as a Hydrophobic Pharmacophore.

Chem. Pharm. Bull. 2000, 48, 312-314.

 

15.    Yamakoshi, Y.; Otani, Y.; Fujii, S.; Endo, Y.*

Dependence of Estrogenic Activity on the Shape of the 4-Alkyl Substituent in Simple Phenols.

Biol. Pharm. Bull., 2000, 23, 259-261.

 

16.    Endo, Y.*; Uchida, T.; Yamaguchi, K.

Anioic [3,3]Rearrangements of Cyclic Hydrazine Diacylates to Medium-size Cyclic Diamides..

Heterocycles, 2000, 53, 151-158.

 

17.    Endo, Y.*; Yokoyama, A.

A. Role of the Hydrophobic Moiety of Protein Kinase C Modulators. Synthesis and Activity of 2-Alkylated Benzolactams

BioMed. Chem. Lett., 2000, 10, 63-66.

 

1999以前

 

18.    Endo, Y.*; Yoshimi, T.; Iijima, T.; Yamakoshi, Y.

Estrogen Antagonists Bearing Dicarba-closo-dodecaborane as a Hydrophobic Pharmacophore.

BioMed. Chem. Lett., 1999, 9, 3387-3392.

 

19.    Endo, Y.*; Iijima, T.; Yamakoshi, Y., Kubo, A.; Itai, A.

Structure-activity Study of Estrogenic Agonists Bearing Dicarba-closo-dodecaborane. Effect of Geometry and Separation Distance of Hydroxyl Groups at the Ends of Molecules.

BioMed. Chem. Lett., 1999, 9, 3313-3318.

 

20.    Endo, Y.*; Taoda, Y.

Electronic Effects of Dicarba-closo-dodecaboranes. Friedel-Crafts Acylation of 1-Phenyl-closo-dodecaboranes.

Tetrahedron Lett, 1999, 40, 9073-9076.

 

21.    Yaguchi, K.; Endo, Y.*

Steric Effects of Polymethyl-dicarba-closo- dodecaboranes. Unusual Reactivity of N-(Deca-B-methyl-1,12-dicarba-closo-dodecaboran-1-carbonyl)pyridinium.

Tetrahedron Lett.,  1999, 40, 7351-7354.

 

22.    Endo, Y.*; Yoshimi, T.; Kimura, K.; Itai, A.

Protein Kinase C Modulators Bearing Dicarba-closo-dodecaborane as a Hydrophobic Pharmacophore.

BioMed. Chem. Lett., 1999, 9, 2561-2564.

 

23.    Endo, Y.*; Iijima, T.; Yamakoshi, Y.; Yamaguchi, M.; Fukasawa, H.; Shudo, K. 

Potent Estrogen Agonists Bearing Dicarba-closo-dodecaborane As a Hydrophobic Pharmacophore.

J. Med. Chem., 1999, 42, 1501-1504.

 

24.    Endo, Y.*; Yaguchi, K.; Tsuji, M.; Shudo, K.

Functionalization of Polymethylcarboranes.  Preparation and Reactivity of Daca-B-methyl-1,12-dicarba-closo-dodecaborane-1-carboxylic Acid.

Chem. Pharm. Bull., 1999, 47, 699-701.

 

25.    Endo, Y.*; Iijima, T.; Ohta, K.; Kagechika, H.; Kawachi, E.; Shudo, K.

Dicarba-closo-dodecaboranes as a Pharmacophore.  Nonel Potent Retinoidal Agonistis.

Chem. Pharm. Bull., 1999, 47, 585-587.

 

26.    Iijima, T.; Endo, Y.*; Tsuji, M.; Kawachi, E.; Kagechika, H.; Shudo, K.

Dicarba-closo-dodecaboranes as a Pharmacophore.  Retinoidal Antagonists and Potential Agonists.

Chem. Pharm. Bull., 1999, 47, 398-404.

 

27.    Kimura, K.; Mizutani, M. Y.; Tomioka, N.; Endo, Y.; Shudo, K.; Itai, A.

Docking Study of Bryostatins to Protein Kinase Cd Cys2 Domain.

Chem Pharm. Bull., 1999, 47, 1134-1137.

 

28.    Endo, Y.*; Shimazu, M.; Fukasawa, H.; Driedger, P. E.; Kimura, K.; Tomioka, N.; Itai, A.; Shudo, K.

Synthesis, Computer Modeling and Biological Evaluation of Novel Protein Kinase C Aginists Based on a 7-Membered Lactam Moiety. 

BioMed. Chem. Lett., 1999, 9, 173-178.

 

29.    Endo, Y.*; Takehana, S.; Ohno, M.; Driedger, P. E.; Stabel, S.; Mizutani, M.; Tomioka, N.; Itai, A.; Shudo, K.

Clarification of the Binding Mode of Teleocidin and Benzolactams to the Cys2 Domain of Protein Kinase Cd by Synthesis of Hydrophobically Modified, Teleocidin-mimicking Benzolactams and Computational Docking Simulation. 

J. Med. Chem., 1998, 41, 1476-1496.

 

30.    Okabe, S.; Sueoka, N.; Komori, A.; Suganuma, M.; Endo, Y.; Shudo, K.; Fujiki, H.

Twist form of Teleocidin Derivatives is Active in in vivo Tumor Promotion by (-)-Benzolactam-V8-310.

Biol. Pharm. Bull., 1998, 21, 465-468.

 

31.    Endo, Y.*; Hirano, M.; Driedger, P. E.; Stabel, S.; Shudo, K.

A Novel Conformational Constrained Analogues of Diacylglycerol. Protein Kinase C Affinity of Simplified Compounds Based on 6-Membered Lactam Moiety.

BioMed. Chem. Lett., 1997, 7, 2997-3000.

 

32.    Yamaguchi, M.; Endo, Y.*; Shimizu, M.; Yamamoto, K.; Yamada, S.; Shudo, K.

3b,5a-Dihydroxycholestan-6-one Exists in Human Blood. 

Biol. Pharm. Bull., 1997, 20, 1044-1046.

 

33.    Endo, Y.*; Uchida, T.; Shudo, K.

Anionic [3,3], [2,3] and [1,2]Rearrangements of Aliphatic and Aromatic Acyl Hydrazines with N-N Bond Cleavage.

Tetrahedron Lett., 1997, 38, 2113-2116.

 

34.    Endo, Y.*; Ohno, M.; Takehana, S.; Driedger, P. E.; Stabel, S.; Shudo, K. 

Role of the Hydrophobic Moiety of Tumor Promoters.  Synthesis and Activity of Benzolactams with Alkyl Substituents at Various Positions. 

Chem. Pharm. Bull., 1997, 45, 424-426.

 

35.    Azuma, A.; Hashimoto, Y.; Yamaguchi, M.; Takehana, S.; Ando, Y.; Iwasaki, S.; Fukasawa, H.; Endo, Y.; Shudo, K.

Photoaffinity Labeling and Affinity Sorbent Gels of Tumor Promoter-Binding Protein (CN-TPBP).

Biol. Pharm. Bull., 1997, 20, 5-8.

 

36.    Shimazu, M.; Endo, Y.*; Shudo, K.

Reactivity of 1,3-Di-t-butylaziridinones with Phenyl Substituents.   A New Fragmentation of a-Lactam. 

Heterocycles, 1997, 735-744.

 

37.    Itai, A.; Matsuo, A.; Mizutani, M.; Tomioka, N.; Endo, Y.; Shudo, K.

Advanced Docking of Two Teleocidin Congeners with the cys2 Domain of Protein Kinase Cd.

Chem. Pharm. Bull., 1997, 45, 573-575.

 

38.    Endo, Y.*; Ohno, M.; Hirano, M.; Itai, A.; Shudo, K.

Synthesis, Conformation and Biological Activity of Teleocidin Mimics, Benzolactams.   A Clarification of the Conformatioal Flexibility Problem in Structure-activity Studies of Teleocidins.     

J. Am. Chem. Soc., 1996, 118, 1841-1855.

 

39.    Endo, Y.*; Yamaguchi, M.; Hirano, M.; Shudo, K. 

Role of the Hydrophobic Moiety of Tumor Promoters.  Synthesis and Activity of 9-Alkylated Benzolactams. 

Chem. Pharm. Bull., 1996, 44,  1138-1140.

 

40.    Matsushima, Y.; Fukasawa, H.; Endo, Y.; Hashimoto, Y.; Shudo K.

Enhancement of Human Papillomavirus Type 18 Gene Expression in Hela Cells by 12-O-Tetradecanoylphorbol-13-acetate, 3b,5a-Dihydroxycholestan- 6-one, and Cholesterol. 

Biol. Pharm. Bull., 1994, 17: 1292-1295.

 

41.    Endo, Y.*; Imada, T.; Yamaguchi, K.; Shudo, K.

Conformational States of Indolactams. Structures of 13-N-Desmethylindolactam-V and 13-O-Indolactam-V.

Heterocycles, 1994, 39: 571-579.

 

42.    Endo, Y.*; Ohno, M.; Hirano, M.; Fujiwara, T.; Sato, A.; Hinuma, Y.; Shudo, K.

Teleocidins and Benzolactams Inhibit Cell Killing by Human Immunodeficiency Virus Type 1 (HIV-1).

Biol. Pharm. Bull., 1994, 17: 1147-1149.

 

43.    Endo, Y.*; Hashimoto, Y.; Fukasawa, H.; Shudo, K.

Synthesis of Oxygenated Cholesterols as Structural Mimics of Phorbol Ester-type Tumor Promoters.

Chem. Pharm. Bull., 1994, 42, 462-469.

 

44.    Endo, Y.*; Ohno, M.; Hirano, M.; Takeda, M.; Itai, A.; Shudo, K.

Chiral Requirement for the Tumor Promoters.  Conformationand Activity Study of Benzolactams.

BioMed. Chem. Lett., 1994, 4, 491-494.

 

45.    Endo, Y.*; Uchida, T.; Hizatate, S.; Shudo, K.

Anionic Hetero [3,3]- and [3,5]Rearrangements of Hydroxylamine Derivatives Accompanied with N-O Bond Cleavage.

Synthesis, 1994, 1096-1105.

 

46.    Endo, Y.*; Uchida, T.; Hizatate, S.; Shudo, K.

Anionic Hetero[3,3] rearrangements of N,O-Diacylhydroxyl- amines to Succinic Acid Derivatives.

Chem. Pharm. Bull., 1994, 42, 419-421.

 

47.    Ohno, M.; Endo, Y.*; Hirano, M.; Itai, A.; Shudo, K.

Designed Molecules Reproducing the Two Conformations of Teleocidins.

Tetrahedron Lett., 1993, 34, 8119-8122.

 

48.    Kawai, T.; Endo, Y.; Yamaguchi, K.; Shudo, K.; Itai, A.

A Crystal Structures of Two Indolactams.

Acta Crystall. 1993, B49: 769-773.

 

49.    Endo, Y.; Hashimoto, Y.; Fukasawa, H.; Shudo, K.

Oxygeneted Steroids as Ligands for Cytosolic-nuclear Tumor Promoter Binding Protein (CN-TPBP).

Biochem. Biophys. Res. Commun., 1993, 193: 1529-1534.

 

50.    Nagata, R.; Endo, Y.*; Shudo, K.

Photocyclization of g-Chlorotiglyl-L-tryptophan Methyl Ester Yields Azocinoindole and Azepinoindole derivatives.

Chem. Pharm. Bull., 1993, 41, 369-372.

 

51.    Paquette, L. A.; Deaton, D. N.; Endo, Y.; Poupart, M-A.

Studies Directed toward the Total Synthesis of Cerorubenic Acid-III. 3. A Convergent Enantioselective Approach Involving New Arrangements for Actuation of Ring D Cyclization.

J. Org. Chem., 1993, 58: 4262-4273.

 

52.    Kawai, T.; Ichinose, T.; Takeda, M.; Tomioka, N.; Endo, Y.; Yamaguchi, K.; Shudo, K.; Itai,A.

Prediction of Ring Conformations of Indolactams. Crystal and Solution Structures. 

J. Org. Chem., 1992, 57, 6150-6155.

 

53.    Kawai, T.; Ichinose, T.; Endo, Y.; Shudo, K.; Itai, A.

Active Conformation of a Tumor Promoter, Teleocidin.  A Molecular Dynamic Study. 

J. Med. Chem., 1992, 35, 2248-2253.

 

54.    Endo, Y.*; Kataoka, K.; Haga, N.; Shudo, K.

Acid-Catalyzed Rearrangement of O-(2-Arylphenyl)hydroxylamines to Aryldihydro-azepinones.

Tetrahedron Lett., 1992, 33, 3339-3342.

 

55.    Haga, N.; Endo, Y.*; Kataoka, K.; Yamaguchi, K.; Shudo, K.

Acid-Catalyzed Amino-Migration of O-Phenylhydroxylamines.

J. Am. Chem. Soc., 1992, 114, 9795-9806.

 

56.    Endo, Y.*; Shudo, K.

Anionic Hetero[3,3]rearrangements.  N-Acyl-N'-enyl-hydrazines to Pyrrolidinines.

Heterocycles, 1992, 33, 91-95.

 

57.    Endo, Y*.; Hizatate, S.; Shudo, K.

Anionic Hetero[3,3]rearrangements. N-Acylhydroxyl-amine-O-carbamates to a-Amino Acids.  A New Method for Introduction of Amino Groups at the a-Position of Carboxylic Acids.

Synlett, 1991, 649-651.

 

58.    Endo, Y.*; Shudo, K.

Anionic 3,4-Diaza[3,3]sigmatropic rearrangements of N,N- Diacyl-hydrazines.

Tetrahedron Lett., 1991, 32: 4517-4520.

 

59.    Endo, Y.*; Hizatate, S.; Shudo, K.

Anionic [3,3]Rearrangement of N-Phenyl-O-acylhydroxyl-amines to o-Aminophenylacetic Acids.

Tetrahedron Lett., 1991, 32: 2803-2806.

 

60.    Itai, A.; Kato, Y.; Tomioka, N.; Iitaka, Y.; Endo, Y.; Hasegawa, M.; Shudo, K., Fujiki, H.; Sakai, S.

A Receptor Model for Tumor Promoters: Rational Superposition of Teleocidins and Phorbol Esters.

Proc. Natl. Acad. Sci. USA., 1988, 85: 3688-3692.

 

61.    Hirota, M.; Suttajit, M.; Endo, Y.; Shudo, K.; Wongchai, V.; Hecker, E.; Fujiki, H.

A New Promoter from the Seed Oil of Jatropha Curcas L.,  An Intramolecular Diester of 12-Deoxy-16-hydroxyphorbol.

Cancer Res., 1988, 48: 5800-5804.

 

62.    Hashimoto, Y.; Endo, Y.; Shudo, K.; Aramaki, Y.; Nakajima, T.

Synthesis of Spider Toxin  and its derivatives.

Pept. Chem. 1988, 363-366.

 

63.    Shudo, K.; Endo, Y.; Aramaki, Y.; Kawai, N.; Nakajima, T.

Newly Synthesized Analogues of the Spider Toxin Block the Crustacean Glutamate Receptor.

Neurosci. Res., 1987, 5: 82-85.

 

64.    Hirota, M.; Suganuma, M.; Yishizawa, S.; Horiuchi, T.; Nakayasu, M.; Hasegawa, M.; Endo, Y.; Shudo, K.; Fujiki, H.

Synthetic Analogues (Indolactams) of Indolactam-V Are New Congeners of the Teleocidin Class Tumor Promoters.

Jpn. J. Cancer Res. (Gann), 1987, 78: 577-582.

 

65.    Endo, Y.; Hasegawa, M.; Itai, A.; Shudo, K.

Synthesis and Stereochemistry of Indolactam Congeners.  Conformational Behavior of the Nine-membered Lactams.

Tetrahedron, 1987, 43: 3695-3704.

 

66.    Hashimoto, Y.; Endo, Y.; Shudo, K.; Aramaki, Y.; Nakajima, T.; Kawai, N.

Synthesis of Spider Toxin (JSTX-3) and Its Analogs.

Tetrahedron Lett., 1987, 28: 3511-3514.

 

67.    Endo, Y.; Sato, Y.; Shudo K.

Synthesis of 7-Substituted Indolactam-V.  An Introduction of Hydrophobic Moeties on the Indole Ring.

Tetrahedron, 1987, 43: 2241-2247.

 

68.    Sakai, S.; Hitotsuyanagi, Y.; Yamaguchi, K.; Aimi, N.; Ogata, K.; Kuramochi, T.; Seki, H.; Hara, R.; Fujiki, H.; Suganuma, M.; Sugimura, T.; Endo, Y.; Shudo, K.; Koyama, Y.

The Structures of Additional Teleocidin Class of Tumor Promoters.

Chem. Pharm. Bull., 1986, 34: 4883-4886.

 

69.    Sakai, S.; Hitotsuyanagi, Y.; Aimi, N.; Fujiki, H.; Suganuma, M.; Sugimura, T.; Endo, Y.; Shudo, K.

Absolute Configuration of Lyngbyatoxin A (Teleocidin A-1) and Teleocidin A-2.

Tetrahedron Lett., 1986, 27: 5219-5220.

 

70.    Endo, Y.; Shudo, K.; Itai, A.; Hasegawa, M.; Sakai, S.

Synthesis and Stereochemistry of Indolactam-V, an Active Fragment of Teleocidins.  Structural Requirement for Tumor-promoting Activity.

Tetrahedron, 1986, 42: 5905-5924.

 

71.    Ninomiya, M.; Fujiki, H.; Paik, N. S.; Hakii, H.; Suganuma, M.; Hitotsuyanagi, Y.; Aimi, N.; Sakai, S.; Endo, Y.; Shudo, K., Sugimura, T.

Des-O-methylolivoretin C Is a New Memberof the Teleocidin Class of Tumor Promoters.

Jpn. J. Cancer Res. (Gann), 1986, 77:  222-225.

 

72.    Endo, Y.; Nanikawa, K.; Shudo, K.

Chemistry of O-Arylhydroxylamines. A Novel Acid-catalyzed Rearrangement of O-Aryl-N-acetoacetylhydroxylamines to Benzofuranes.

Tetrahedron Lett., 1986, 27: 4209-4212.

 

73.    Endo, Y.; Hasegawa, M.; Itai, A.; Shudo, K.; Tori, M.; Asakawa, Y.; Sakai, S.

Tumor promoters Exist in Two Conformational States in Solution.  Stereochemistry of Indolactam-V.

Tetrahedron Lett., 1985, 26: 1069-1072.

 

74.    Fujiki, H.; Suganuma, M.; Hakii, H.; Nakayasu, M.; Endo, Y.; Shudo, K.; Irie, K.; Koshimizu, K.; Sugimura, T.

Tumor Promoting activities of New Synthetic Analogues of Teleocidin.

Pro. Japan. Acad.(B), 1985, 61: 45-48.

 

75.    Hitotsuyanagi, Y.; Fujiki, H.; Suganuma, M.; Aimi, N.; Sakai, S.; Endo, Y.; Shudo, K.; Sugimura, T.

Isolation and Structure Elucidation of Teleocidin B-1, B-2, B-3 and B-4.

Chem. Pharm. Bull., 1984, 32: 4233-4236.

 

76.    Hitotsuyanagi, Y.; Yamaguchi, K.; Ogata, K.; Aimi, N.; Sakai, S.; Koyama, Y.; Endo, Y.; Shudo, K.; Itai, A.; Iitaka, Y.

Elucidation of the Structures of Olivoretin B and C.

Chem. Pharm. Bull., 1984, 32: 3774-3778.

 

77.    Horiuchi, T.; Fujiki, H.; Suganuma, M.; Hakii, H.; Nakayasu, M.; Hitotsuyanagi, Y.; Aimi, N.; Sakai, S.; Endo, Y.; Shudo, K.; Sugimura, T.

Studies on Olivoretins Indicate a Requirment for a Free Hydroxyl Group for Teleocidin B Activity.

Jpn. J. Cancer Res. (Gann), 1984, 75: 837-840.

 

78.    Fujiki, H.; Suganuma, M.; Nakayasu, M.; Tahira, T.; Endo, Y.; Shudo, K.; Sugimura, T.

Structure Activity Studies on Synthetic Analogues (Indolactams) of the Tumor Promoter Teleocidin.

Jpn. J. Cancer Res. (Gann), 1984, 75: 866-870.

 

79.    Endo, Y.; Shudo, K.; Furuhata, K.; Ogura, H.; Sakai, S.; Aimi, N.; Hitotsuyanagi, Y.; Koyama, Y.

Synthesis of Optically Active Teleocidin Derivatives.  Absolute Configuration of Teleocidin B and Olivoretin A.

Chem. Pharm. Bull., 1984, 32: 358-361.

 

80.    Endo, Y.; Terashima, T.; Shudo, K.

A Novel Acid-catalyzed Rearrangement of N-Aryl-N'-aryloxyureas to Biphenyl Derivatives. A [5,5]Rearrangement Involving Three Heteroatoms.

Tetrahedron Lett., 1984, 25: 5537-5540.

 

81.    Iijima, H.; Endo, Y.; Shudo, K.; Okamoto, T.

Phenoxenium Ions. Identical Intermediates in the Acid-catalyzed Solvolysis of N-Tosyl-O-arylhydroxylamines and in the Thermolysis of N-aryloxypyridinium Salts.

Tetrahedron, 1984, 40: 4981-4985.

 

82.    Endo, Y.; Shudo, K.; Okamoto, T.

An Acid Catalyzed Rearrangement of N-Alkyl-N'-phenoxyureas; Synthesis of 2-Alkylaminophenols from Phenols.

Synthesis, 1983, 471-473.

 

83.    Endo, Y.; Shudo, K.; Okamoto, T.

Formation of Punmerer's Ketone from 4-Methylphenoxenium Ion. An Acid-catalyzed Solvolysis of N-p-Toluenesulfonyl-O-(4-tolyl)hydroxylamine in p-Cresol.

Chem. Pharm. Bull., 1983, 31: 3769-3770.

 

84.    Endo, Y.; Shudo, K.; Okamoto, T.

Molecular Requirements for epigenetic Modulators. Synthesis of Active Fragment of Teleocidins and Lyngbyatoxin.

Chem. Pharm. Bull., 1982, 30: 3457-3460.

 

85.    Endo, Y.; Shudo, K.; Okamoto, T.

An Acid-catalyzed Solvolysis of N-Sulfonyl- and N-Acylhydroxylamines; Phenoxenium Ions.

J. Am. Chem. Soc., 1982, 104: 6393-6397.

 

86.    Endo, Y.; Shudo, K.; Okamoto, T.

Reaction of Benzene with Diphenylsulfoxides.

Chem. Pharm. Bull., 1981, 29: 3753-3755.

 

87.    Endo, Y.; Shudo, K.; Okamoto, T.

An Acid Catalyzed Rearrangement of O-Aryl-N-benzoylhydroxylamines: Synthesis of Catechols from Phenols.

Synthesis, 1980, 461-463.

 

88.    Ohta, T.; Machida, R.; Takeda, K.; Endo, Y.; Shudo, K.; Okamoto, T.

Reductive Phenylation of Nitroarenes.

J. Am. Chem. Soc., 1980, 102: 6385-6386.

 

89.    Endo , Y.; Shudo, K.; Okamoto, T.

A Novel Phenol-benzene Coupling Reaction. An Acid-catalyzed Reaction of N-Acyl-O-arylhydroxylamines with Benzene.

J. Am. Chem. Soc., 1977, 99: 7721-7723.

 

90.    Endo, Y.; Ohta, T.; Shudo, K.; Okamoto, T.

Reaction of Arylhydroxamic Acids with Benzene.

Heterocycles, 1977, 8: 367-370.

 

91.    Shudo, K.; Ohta, T.; Endo, Y.; Okamoto, T.

Phenylation of N,N-Dialkylaniline-N-oxides.

Tetrahedron Lett., 1977, 18: 105-108.

 

総説

 

92.    太田公規:超分子化学を利用した創薬:麻酔剤の使用法に革命を起こすホスト化合物

ファルマシア 2013, 49, 444

 

93.    太田公規, 遠藤泰之:ホウ素クラスターを用いた実践的創薬研究

ファルマシア 2012, 48, 504-508.

 

94.    遠藤泰之, 太田公規: ホウ素クラスター:カルボランの有機化学―合成、構造、立体分子構築への応用

有機合成化学協会誌, 2007, 65: 320-333.

 

95.    遠藤泰之ホウ素クラスターの医薬化学の医薬化学への応用

東北薬科大学研究誌, 2003, 50: 1-16.

 

96.    遠藤 泰之: ホウ素クラスターの医薬化学への応用:カルボラン骨格を有するエストロゲン受容体リガンド、

MEDCHEM NEWS (DISCOVERY), 2000, 10: No 3. 20-24.

 

97.    遠藤 泰之: ホウ素クラスターの医薬化学

         現代化学, 1999, 342: 51-58.

 

98.    遠藤 泰之: 発がんプロモーターの活性立体構造の解析、

         RADIOISOTOPES, 1996, 45: 95-104.

 

99.    遠藤 泰之、大野 道博、首藤 紘一: テレオシジンの活性立体配座:新規活性分子のデザインと合成、

         薬学雑誌、総説(総合論文)1994, 114:  464-477.

 

100.遠藤 泰之、首藤 紘一: フェノキセニウムイオンの生成と反応、

         薬学雑誌、総説(総合論文)1994, 114:  565-576.

 

101.遠藤 泰之: 発癌プロモーター、テレオシジンの合成と生物活性、

         有機合成化学協会誌、1988, 46: 344-355.

 

102.遠藤 泰之: Teleocidin を含むTPAタイプのプロモーターの活性構造の解析、

         日本農芸化学会誌、1987, 61: 834-837.

 

103.遠藤 泰之、板井 昭子、首藤 紘一、藤木 博太: 発がんプロモーターの活性構造、

         癌と化学療法、1986, 13: 3365-3375.

 

104.藤木 博太、菅沼 雅美、遠藤 泰之、首藤 紘一ら: TPAタイプおよび non-TPAタイプ発癌プロモーターの活性と作用機構、

         癌と化学療法、1986, 13: 758-765.

 

単行書

 

105.Endo, Y. Carboranes as Hydrophobic Pharmacophores: Applications for Design of Nuclear Receptor Ligands “Boron-Based Compounds: Potential and Emerging Applications in Medicine”, Evamarie Hey-Hawkins, E., Vinas, C. (eds.), Wiley-VHC, Weinheim, pp3-19, 2018.

 

106.Endo, Y.; Yoshimi, T.; Miyaura, C: Utility of Boron Cluster for Drug Design: Selective Estrogen Receptor Modulators (SERMs) Bearing Carborane As a Hydrophobic Skeletal Structure., “Boron Chemistry at the Beginning of the 21th century”, Bubnov, Yu., et al (eds.), Russian Academy of Sciences, Nauka, Moscow, pp298-306, 2003.

 

107.Gabel, D.; Endo, Y.: Polyboranes in Medicinal Chemistry. “Molecular Clusters of the Main-Group Elements”, Driess, M.; Noth, H (eds.), Wiley-VHC, Weinheim, 2003.

 

108.遠藤泰之: 受容体の構造と細胞内情報伝達(訳), “オックスフォード・メディシナルケミストリー”, 北川勲、柴崎正勝、富岡清 監訳 (p91-118) 丸善(東京), 2003.

 

109.Endo, Y*.: A New Medicinal Application of Boron Clusters. Potent Nuclear Receptor Ligands Bearing Carborane as a Hydrophobic Pharmacophore.

“Contemporary Boron Chemistry”, Wade, K., et al (eds.), the Royal Society of Chemistry, Cambridge Science Press, Cambridge, pp139-143, 2000.

 

110.遠藤 泰之*: 発癌プロモーター、テレオシジンの化学と生物活性,

         発癌と制癌の化学(p83-114)  廣川書店(東京), 1990.

 

111.Fujiki, H., Suganuma, M., Tahira, T., Yoshioka, A., Nakayasu, M., Endo, Y., Shudo, K., Takayama, S., Moore, R. E., Sugimura, T.: New Classes of Tumor Promoters: Teleocidin, Aplysiatoxin and Palytoxin., 

"Cellular Interactions by Environmental Tumor promoters" Fujiki,H., et al (eds.), Japan Sci. Soc. Press, Tokyo/ VNU Science Press, Utrecht, pp37-45, 1984.

 

教科書

 

112.遠藤泰之、スタンダード薬学シリーズU 化学系薬学 II 生体分子・医薬品の化学による理解(日本薬学会編)東京化学同人(東京)2016, p186-191, 6/ 337

 

113.遠藤泰之、スタンダード薬学シリーズ 化学系薬学 I 化学物質の性質と反応(日本薬学会編)東京化学同人(東京)2015, p360-369, 10/ 437

 

114.遠藤泰之、スタンダード薬学シリーズ 化学系薬学 IV 演習編(日本薬学会編)東京化学同人(東京)2008, p107-112, p116-117, 8/204

 

115.遠藤泰之、ベーシック薬学教科書シリーズ 創薬科学・医薬化学、(橘高敦史編)

        化学同人(京都) 2007, p165-216, 52/297                                                                                

116.遠藤泰之、知っておきたい有機反応100(日本薬学会編)        

        東京化学同人(東京)2006, p47-62, 16/254  

 

117.遠藤泰之、スタンダード薬学シリーズ 化学系薬学 II ターゲット分子の合成と生体分子・医薬品の化学(日本薬学会編)東京化学同人(東京)2005, p184-190, 7/240                           

118.遠藤泰之「創薬科学 生体構成分子から見た医薬品」(石橋弘行編) 

        廣川書店(東京) 2004, p1-14, p37-54, p88-98, 43/192

 

119.遠藤泰之、スタンダード薬学シリーズ 化学系薬学 I 化学物質の性質と反応(日本薬学会編)東京化学同人(東京)2004, p216-220, 5/ 327

 

120.遠藤泰之、スタンダード薬学シリーズ 医薬品の開発と生産(日本薬学会編)

東京化学同人(東京)2004, p81-90, 10/ 212

 


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