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発表論文JOURNAL

2020~

2026年

The protective function of TRPV4 in interstitial cystitis/bladder pain syndrome.
Masaru Yoshizumi
Yakugaku Zasshi., 146: 157-163, 2026

2025年

Characterizations of actions of the novel gabapentinoid drug mirogabalin on painful bladder hypersensitivity in rats with lipopolysaccharide-induced chronic cystitis.
Masaru Yoshizumi, Yutaka Kitano, Chizuko Watanabe, Shinobu Sakurada, Hirokazu Mizoguchi.
Life Sci., 380: 123942, 2025

2024年

Characteristics of α1-adrenoceptor antagonists-induced ejaculatory dysfunction on spontaneous seminal emission in rats.
Masaru Yoshizumi, Shin-nosuke Ise, Akihiko Yonezawa, Chizuko Watanabe, Shinobu Sakurada, Hirokazu Mizoguchi.
Basic Clin. Pharmacol. Toxicol., 134: 704-711, 2024

2022年

TRPV4 activation prevents lipopolysaccharide-induced painful bladder hypersensitivity in rats by regulating immune pathways.
Masaru Yoshizumi, Naoya Tazawa, Chizuko Watanabe, Hirokazu Mizoguchi.
Front. Immunol., 13: 1080302, 2022

Translational value of the transdermal administration of bergamot essential oil and of its fractions.
Damiana Scuteri, Laura Rombola, Michele Crudo, Chizuko Watanabe, Hirokazu Mizoguchi, Shinobu Sakurada, Kengo Hamamura, Tsukasa Sakurada, Luigi Antonio Morrone, Paolo Tonin, Giacinto Bagetta, Maria Tiziana Corassaniti.
Pharmaceutics., 14: 1006, 2022

Preclinical characterization of antinociceptive effect of bergamot essential oil and of its fractions for rational translation in complementary therapy.
Damiana Scuteri, Laura Rombola, Michele Crudo, Chizuko Watanabe, Hirokazu Mizoguchi, Shinobu Sakurada, Kengo Hamamura, Tsukasa Sakurada, Paolo Tonin, Maria Tiziana Corassaniti, Giacinto Bagetta.
Pharmaceutics., 14: 312, 2022

Synthesis of unnatural morphinan compounds to induce itch-like behaviors in mice: Towards the development of MRGPRX2 selective ligands.
Keita Ito, Noriki Kutsumura, Yasuyuki Nagumo, Tsuyoshi Saitoh, Akihisa Tokuda, Kao Hashimoto, Naoshi Yamamoto, Ryoji Kise, Asuka Inoue, Hirokazu Mizoguchi, Hiroshi Nagase.
Bioorg. Med. Chem. Lett., 56: 128485, 2022

2021年

Development and translation of nanoBEO, a nanotechnology-based delivery system of bergamot essential oil deprived of furocumarins, in the control of agitation in severe dementia.
Damiana Scuteri, Rosaria Cassano, Sonia Trombino, Rossella Russo, Hirokazu Mizoguchi, Chizuko Watanabe, Kengo Hamamura, Soh Katsuyama, Takaaki Komatsu, Luigi Antonio Morrone, Laura Rombola, Annagrazia Adornetto, Annarita S. Lagani, Maria Tiziana Corassaniti, Paolo Tonin, Shinobu Sakurada, Tsukasa Sakurada, Pierluigi Nicotera, Giacinto Bagetta.
Pharmaceutics., 13: 379, 2021

Gabapentin reduces painful bladder hypersensitivity in rats with lipopolysaccharide-induced chronic cystitis.
Masaru Yoshizumi, Chizuko Watanabe, Hirokazu Mizoguchi.
Pharmacol. Res. Perspect., 9: e00697, 2021

Central mechanisms of apomorphine and m-chlorophenylpiperazine on synergistic action for ejaculation in rats.
Masaru Yoshizumi, Akihiko Yonezawa, Yukio Kimura, Chizuko Watanabe, Shinobu Sakurada, Hirokazu Mizoguchi.
J. Sex. Med., 18: 231-239, 2021

2020年

Exploring μ-opioid receptor splice variants as specific molecular target for new analgesics.
Hirokazu Mizoguchi, Hideaki Fujii.
Curr. Top. Med. Chem., 20: 2866-2877, 2020

Morphine antinociception restored by use of methadone in the mophine-resistant inflammatory pain state.
Chizuko Watanabe, Asami Komiyama, Masaru Yoshizumi, Shinobu Sakurada, Hirokazu Mizoguchi.
Front. Pharmacol., 11: 593647, 2020

Effectiveness of gabapentinoids for cancer-related rectal and vesical tenesmus: Report of four cases.
Keita Tagami, Masaru Yoshizumi, Akira Inoue, Motohiro Matoba.
Indian. J. Palliat. Care., 26: 381-384, 2020

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